Linagliptin

Product Description:

Product Name: Linagliptin CAS NO:668270-12-0

Synonyms:

(R)-8-(3-aminopiperidin-1-yl)-7-(but-2-yn-1-yl)-3-Methyl-1-((4-Methylquinazolin-2-yl)Methyl)-1H-purine-2,6(3H,7H)-dione;

Chemical & Physical Properties:

Appearance : White or off-white crystalline powder

Assay : No less than 99%

Melting point: 202℃

Density: 1.39/cm³

Boiling point: 661.189℃

Flash point: 353.675℃

Vapour Pressure: 0.0±2.0 mmHg at 25°C

Index of Refraction: 1.717

Category: Pharmaceutical raw material; Inhibitor;Amines;Aromatics;Heterocycles;Intermediates & Fine Chemicals; Pharmaceutical API.

Safety Information:

Safety Statements: S36/37

Risk Statements: R20/21/22

Hazard Codes: Xi

HS Code: 2933590090

Storage:Stored in a cool and dry well-closed container. Keep away from moisture and strong light/heat.

Application: 

1.Linagliptin(BI-1356) is an inhibitor of DPP-4, an enzyme that degrades the incretin hormones glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP).

2. 8-[(3R)-3-Amino-1-piperidinyl]-7-(2-butyn-1-yl)-3-methyl-1-[(4-methyl-2-quinazolinyl)methyl]-3,7-dihydro-1H-purine-2,6-dione is an novel potent and selective dipeptidyl peptidase-4 (DPP-4) inhibitor with potential use in the treatment of type 2 diabetes.

Our factory manufacture’s Linagliptin CAS 668270-12-0, mature technology, stable output, quality assurance.

Inventory Status : In Stock.

We can provide (R)-8-(3-aminopiperidin-1-yl)-7-(but-2-ynyl)-3-methyl-1-((4-methylquinazolin-2-yl)methyl)-1H-purine-2,6(3H,7H)-dione certificate of analysis( COA), 8-[(3R)-3-aminopiperidin-1-yl]-7-but-2-ynyl-3-methyl-1-[(4-methylquinazolin-2-yl)methyl]purine-2,6-dione MOA, 1H-Purine-2,6-dione,8-[(3R)-3-aMino-1-piperidinyl]-7-(2-butyn-1-yl)-3,7-dihydro-3-Methyl-1-[(4-Methyl-2-quinazolinyl)Methyl]- ROS, Linagliptin CAS 668270-12-0 MSDS and other support for you !

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